Exemestane

Description

Common names in USA Aromadex, Aromasin, Aromaxyl. Description of the drug Yellow round pills of compact and homogeneous structure. Aromamine composition 1 tablet contains: Active substance: Exemestane 25mg Benefits of bodybuilding Aromasin (Exemestane) – a new generation of drugs that blocks the enzymes responsible for aromatization. Exemestane is significantly different from drugs belonging to the class of aromatase inhibitors. In USA Aromasin is a better drug. Familiar aromatase inhibitors have only temporary effectiveness, but Aromasin has an irreversible and permanent effect. Due to the drugs are suppressed 85% or more of estrogen in the athlete's body. Aromasin during the steroid cycle prevents the side effects that steroids can cause – aroma. It should be noted that the effect of Aromasin is fundamentally different from the usual action of Nolvadex for many athletes. It is known that tamoxifen has no effect on the aromatization process. It just begins to interact with cellular estrogen receptors, preventing estrogen from joining them and forming a bond. Exemestane also acts on the aromatization process and suppresses it. The structure of Aromasin is very similar to a natural steroid – androstenedione. The operating principle of exemestane is that it binds irreversibly to hormone-active enzymes. As a result, the hormones lose their activity. Aromasin has no estrogenic or progestogenic activity. But it is characterized by mild androgenic activity. Therapeutic indication Breast cancer in postmenopausal women (natural or induced), progressing against the background of antisterogen therapy, nonsteroidal aromatase inhibitors or progestins. Dosage (Men) 12.5-25mg/day Dosage (Women) 12.5mg/day Active life 9 hours Aromasin Side Effects Aromasin side effects can occur frequently and to varying degrees. For example, an athlete may experience such unpleasant consequences as: nausea, fatigue, sweating, dizziness, headache, rash, insomnia, etc. In one athlete side effects can occur quickly, in others the use of the drug can pass completely painless. It all depends on the individual sensitivity of the man to the active ingredient of the drug. But usually, subject to recommended doses, Aromasin side effects do not appear or occur only to a small extent. Aromasin Contraindications / Precautionary measures in USA Hypersensitivity. Not recommended for women with pre-menopausal endocrine status (the efficacy and safety of the drug in this group of patients has not been studied). In patients with hepatic or renal insufficiency, a dose adjustment is necessary. Do not use in children. During treatment should refrain from activities that require concentration and speed of psychomotor reactions (when using the drug were observed such symptoms as drowsiness, fatigue and dizziness). Overdose Treatment: symptomatic (specific antidote does not exist), regular monitoring of vital signs and careful observation.